Medicinal Chemistry: Course Outline IVB-719

General properties chemistry biological action structure activity relationship and therapeutic applications of following

Sulphonamides

• Prontosil
• Sulphanilamide
• Sulphapyridine
• Sulphadimidine
• Sulfamethoxazole
• Sulfadiazine
• Sulfafurazole​

Antimalarials

• 4-Aminoquinolines
• 8-Aminoquinolines
• 9-Amino acridines
• Biguanides
• Pyrimidine analogues
• Mefloquine
• Cinchona alkaloids

 Diuretics

• Mercaptomerin
• Meralluride
• Thiazides
• Sprironolactone
• Theophylline
• Furosemide
• Acetazolamide
• Ethacrynic acid
• Triameterene

Antitubercular drugs

• Ethambutol
• Isonicotinic acid
• Hydrazid
• Rifampacin
• Thioguanine
• Pyrazinamide
• Cycloserine
• Ethunamide
• Cytarabine
• 5-Flourouracil
• Dacarbazine​

Antiviral drugs

• Acyclovir
• Tromantadine hydrochloride and ribavirin​

Immunosuppressant agents

• Azathioprine and cyclosporin

Antibiotics

• Penicillins
• Cephalosporins
• Streptomycin
• Chloramphenicol
• Tetracyclines
• Kanamycin
• Erythromycin